Sulfoxide-directed stereocontrolled access to 2H-chromans: Total synthesis’ of the (S,R,R,R)-enantiomer of the antihypertensive drug nebivolol

M. C. Carreno, G. Hernandez-Torres, A. Urbano, F. Colobert

Eur. J. Org. Chem. 2008, 2035-2038

Publications

New analogs of polysphorin and uses thereof for treating or preventing malaria

S. Choppin, F. Colobert, G. Hanquet, F. Leroux, D. Mazier, N. Mahmoudi

EP 08 305646.5 (Université Louis Pasteur, CNRS, Assistance Publique – Hôpitaux de Paris, Université Pierre et Marie Curie; 7/10/2008)

Patents

Suzuki-Miyaura Coupling Reaction of Boronic Acids and Ethyl Glyoxylate: Synthetic Access to Mandelate Derivatives

I. N. Francesco, A. Wagner, F. Colobert

Eur. J. Org. Chem. 2008, 5692-5695

Publications

Large-Scale Preparation of Enantiomerically Pure (4aR)-(-)-1,4a-Dimethyl-4,4a,7,8-tetrahydronaphthalene-2,5(3H,6H)-dione: A Useful Wieland-Miescher Diketone Analogue

D. A. Lanfranchi, N. Baldovini, G. Hanquet

Synthesis-Stuttgart 2008, 3775-3778

Publications

Polysubstituted oxygen heterocycles by a Reformatsky-type reaction/reductive cyclization approach from enantiopure beta-ketosulfoxides

F. Colobert, S. Choppin, L. Ferreiro-Mederos, M. Obringer, S. L. Arratta, A. Urbano, M. C. Carreno

Org. Lett. 2007, 9, 4451-4454

Publications

Stereoselective synthesis of the C(53)-C(67) polyene fragment of amphidinol 3

F. Colobert, T. Kreuzer, J. Cossy, S. Reymond, T. Tsuchiya, L. Ferrie, I. E. Marko, P. Jourdain

Synlett 2007, 2351-2354

Publications

Efficient syntheses of the polyene fragments present in amphidinols

J. Cossy, T. Tsuchiya, L. Ferrie, S. Reymond, T. Kreuzer, F. Colobert, P. Jourdain, I. E. Marko

Synlett 2007, 2286-2288

Publications

Relative Carbanion Basicity as Driving Force for an Intramolecular Silyl Migration of Lithiated Biphenyls

L. Bonnafoux, R. Scopelliti, F. R. Leroux, F. Colobert

Tetrahedron Lett. 2007, 48, 8768-8772

Publications

A Practical Transition-metal-free Aryl-Aryl Coupling Method : Arynes as Key Intermediates

F. R. Leroux, L. Bonnafoux, C. Heiss, F. Colobert, D. A. Lanfranchi

Adv. Synth. Catal. 2007, 349, 2705-2713

Publications

Triazolopyridines. Part 25. Synthesis of new chiral ligands from [1,2,3]triazolo[1,5-a]pyridines

B. Abarca, R. Ballesteros, R. Ballesteros-Garrido, F. Colobert, F. R. Leroux

Tetrahedron 2007, 63, 10479-10485

Publications