Archive for 2008

Triazolopyridines. Part 26. The preparation of novel [1,2,3]triazolo[1,5-a]pyridine sulfoxides

B. Abarca, R. Ballesteros, R. Ballesteros-Garrido, F. Colobert, F. R. Leroux

Tetrahedron 2008, 64, 3794-3801


Sulfoxide-directed stereocontrolled access to 2H-chromans: Total synthesis’ of the (S,R,R,R)-enantiomer of the antihypertensive drug nebivolol

M. C. Carreno, G. Hernandez-Torres, A. Urbano, F. Colobert

Eur. J. Org. Chem. 2008, 2035-2038


New analogs of polysphorin and uses thereof for treating or preventing malaria

S. Choppin, F. Colobert, G. Hanquet, F. Leroux, D. Mazier, N. Mahmoudi

EP 08 305646.5 (Université Louis Pasteur, CNRS, Assistance Publique – Hôpitaux de Paris, Université Pierre et Marie Curie; 7/10/2008)


Suzuki-Miyaura Coupling Reaction of Boronic Acids and Ethyl Glyoxylate: Synthetic Access to Mandelate Derivatives

I. N. Francesco, A. Wagner, F. Colobert

Eur. J. Org. Chem. 2008, 5692-5695


Large-Scale Preparation of Enantiomerically Pure (4aR)-(-)-1,4a-Dimethyl-4,4a,7,8-tetrahydronaphthalene-2,5(3H,6H)-dione: A Useful Wieland-Miescher Diketone Analogue

D. A. Lanfranchi, N. Baldovini, G. Hanquet

Synthesis-Stuttgart 2008, 3775-3778